{"id":396912,"date":"2026-08-25T16:57:16","date_gmt":"2026-08-25T16:57:16","guid":{"rendered":"http:\/\/6a8dafba694551c2d98c91f1"},"modified":"2026-08-25T16:57:16","modified_gmt":"2026-08-25T16:57:16","slug":"una-mutacion-amenaza-el-tratamiento-mas-usado-contra-la-malaria","status":"publish","type":"post","link":"https:\/\/sarmiento24h.com\/?p=396912","title":{"rendered":"Una mutaci\u00f3n amenaza el tratamiento m\u00e1s usado contra la malaria"},"content":{"rendered":"<div><img decoding=\"async\" src=\"https:\/\/media.es.wired.com\/photos\/6a8dafba9b6cd8eaf0679e81\/16:9\/w_1280,c_limit\/139813972\" class=\"ff-og-image-inserted\"><\/div>\n<p>Durante muchos a\u00f1os, en el \u00c1frica subsahariana, el f\u00e1rmaco a base de artemisinina \u201cartem\u00e9ter-lumefantrina\u201d se ha usado ampliamente como tratamiento principal para la malaria, una enfermedad infecciosa transmitida por mosquitos. Pero en los \u00faltimos a\u00f1os, ha surgido preocupaci\u00f3n por una disminuci\u00f3n en la susceptibilidad de los par\u00e1sitos de la malaria a este f\u00e1rmaco, lo que hace urgente dilucidar los factores gen\u00e9ticos subyacentes.<\/p>\n<p>Por lo tanto, un equipo de investigaci\u00f3n de la Universidad de Brown realiz\u00f3 un an\u00e1lisis del genoma completo de par\u00e1sitos de la malaria a partir de 157 muestras seleccionadas de espec\u00edmenes recolectados en Uganda entre 2016 y 2024. Buscaron regiones gen\u00e9ticas involucradas en la reducci\u00f3n de la susceptibilidad a los f\u00e1rmacos. Como resultado, <a href=\"https:\/\/www.nature.com\/articles\/s41591-026-04590-5\" target=\"_blank\">encontraron<\/a> rastros de una fuerte selecci\u00f3n natural (el fen\u00f3meno en el que las mutaciones ventajosas para la supervivencia se propagan r\u00e1pidamente) en un gen llamado \u00abpx1\u00bb, que no hab\u00eda recibido mucha atenci\u00f3n hasta entonces.<\/p>\n<p>\u201cLa malaria sigue siendo una de las principales causas de muerte, especialmente en el \u00c1frica subsahariana\u201d, explica Jeffrey Bailey, profesor asociado de patolog\u00eda en la Universidad de Brown. \u201cSi la resistencia a los medicamentos contin\u00faa desarroll\u00e1ndose, ser\u00e1 m\u00e1s dif\u00edcil controlar la propagaci\u00f3n de la infecci\u00f3n, y existe la preocupaci\u00f3n de que muchas personas pierdan la vida tanto dentro como fuera de la regi\u00f3n\u201d.<\/p>\n<h2>Un grupo de mutaciones que se propag\u00f3 r\u00e1pidamente<\/h2>\n<p>Cuando Bailey y su equipo de investigaci\u00f3n examinaron el gen px1 en detalle, descubrieron que se heredaba como un conjunto de tres mutaciones de amino\u00e1cidos y dos deleciones (un fen\u00f3meno en el que se pierde una parte del cromosoma o de la secuencia de bases del ADN). Los investigadores denominaron a este grupo de mutaciones \u00abPIN\u00bb.<\/p>\n<p>Los genes se recombinan con cada generaci\u00f3n y eso provoca una alteraci\u00f3n gradual de su secuencia. Sin embargo, en los par\u00e1sitos de la malaria portadores de la mutaci\u00f3n PIN, una amplia regi\u00f3n alrededor del gen px1 se conserv\u00f3 casi por completo en m\u00faltiples individuos. Esto sugiere que no hab\u00eda transcurrido el tiempo suficiente desde la aparici\u00f3n de la mutaci\u00f3n PIN para que se produjera la \u201crecombinaci\u00f3n gen\u00e9tica\u201d, lo que indica que se propag\u00f3 r\u00e1pidamente en los \u00faltimos a\u00f1os.<\/p>\n<p>Para determinar cu\u00e1ndo apareci\u00f3 por primera vez la mutaci\u00f3n PIN, el equipo de investigaci\u00f3n revis\u00f3 muestras anteriores y la identific\u00f3 inicialmente en una muestra de 2008. Posteriormente, la mutaci\u00f3n PIN se propag\u00f3 a un ritmo asombroso. Se estima que para 2016 en el norte de Uganda y para 2023 en el este, m\u00e1s de la mitad de los par\u00e1sitos de la malaria portaban esta mutaci\u00f3n. Para 2024, hab\u00eda alcanzado el 84% en el norte y el 55% en el este.<\/p>\n<p>Adem\u00e1s, el equipo de investigaci\u00f3n compar\u00f3 la respuesta a los f\u00e1rmacos en individuos con y sin la mutaci\u00f3n PIN en los par\u00e1sitos de la malaria. Los resultados mostraron que los par\u00e1sitos de la malaria con la mutaci\u00f3n PIN respond\u00edan menos a la lumefantrina, un componente de la artem\u00e9ter-lumefantrina, a la dihidroartemisinina, que se produce cuando el otro componente, el artem\u00e9ter, se convierte en el organismo, y a la mefloquina, otro f\u00e1rmaco contra la enfermedad.<\/p>\n<p>Para confirmar si este resultado se deb\u00eda realmente al gen px1, los investigadores usaron par\u00e1sitos de la malaria creados en un estudio anterior mediante la interrupci\u00f3n intencional del gen px1 y examinaron de forma similar su respuesta a los f\u00e1rmacos. Descubrieron que los individuos que carec\u00edan del gen px1 respond\u00edan con mayor intensidad a estos f\u00e1rmacos terap\u00e9uticos.<\/p>\n<p>Esto confirma que el gen px1 influye en la respuesta a los f\u00e1rmacos. Por otro lado, un estudio que investig\u00f3 la resistencia a la artemisinina no hall\u00f3 diferencias claras basadas en mutaciones del gen PIN.<\/p>\n<h2>Nuevas pistas que se suman a la red de vigilancia<\/h2>\n<p>Anteriormente, se sab\u00eda que la resistencia a la artemisinina estaba asociada con mutaciones en el gen Kelch13 (K13). Sin embargo, no se hab\u00edan encontrado mutaciones marcadoras verificadas para la lumefantrina, el otro componente de las combinaciones de f\u00e1rmacos basadas en artemisinina.<\/p>\n<p>Si bien se hab\u00eda sugerido una posible relaci\u00f3n con mutaciones en otros genes, su impacto era m\u00ednimo y no se consideraba un indicador fiable. Este descubrimiento constituye el primer estudio que demuestra que una mutaci\u00f3n en un solo gen puede estar relacionada con una menor sensibilidad tanto al artem\u00e9ter como a la rumefantrina.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Durante muchos a\u00f1os, en el \u00c1frica subsahariana,&#46;&#46;&#46;<\/p>\n","protected":false},"author":1,"featured_media":396913,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"_jetpack_newsletter_access":"","_jetpack_dont_email_post_to_subs":false,"_jetpack_newsletter_tier_id":0,"_jetpack_memberships_contains_paywalled_content":false,"_jetpack_feature_clip_id":0,"_jetpack_memberships_contains_paid_content":false,"footnotes":"","jetpack_publicize_message":"","jetpack_publicize_feature_enabled":true,"jetpack_social_post_already_shared":true,"jetpack_social_options":{"image_generator_settings":{"template":"highway","default_image_id":0,"font":"","enabled":false},"version":2},"jetpack_post_was_ever_published":false},"categories":[46],"tags":[],"class_list":["post-396912","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-tecnologia"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v28.1 - 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